Comment
|
AKT1 interacts with PDPK1.
|
Formal Description Interaction-ID: 1890
|
interacts (colocalizes) with
|
Drugbank entries
|
Show/Hide entries for
AKT1
or
PDPK1
|
Drugbank
DB00171
|
|
Drugbank
DB01169
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB07584
|
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)phe ...
|
Drugbank
DB07585
|
5-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-4 ...
|
Drugbank
DB00171
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB00482
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB01933
|
|
Drugbank
DB01946
|
3-[1-(3-Aminopropyl)-1h-Indol-3-Yl]-4-(1 ...
|
Drugbank
DB02010
|
|
Drugbank
DB03777
|
|
Drugbank
DB04522
|
|
Drugbank
DB06932
|
10,11-dimethoxy-4-methyldibenzo[c,f]-2,7 ...
|
Drugbank
DB07033
|
5-HYDROXY-3-[(1R)-1-(1H-PYRROL-2-YL)ETHY ...
|
Drugbank
DB07132
|
1-{2-OXO-3-[(1R)-1-(1H-PYRROL-2-YL)ETHYL ...
|
Drugbank
DB07300
|
2-(1H-imidazol-1-yl)-9-methoxy-8-(2-meth ...
|
Drugbank
DB07456
|
3-(1H-INDOL-3-YL)-4-(1-{2-[(2S)-1-METHYL ...
|
Drugbank
DB07457
|
3-[1-(3-AMINOPROPYL)-1H-INDOL-3-YL]-4-(1 ...
|
Drugbank
DB00482
|
|
Drugbank
DB01933
|
|
Drugbank
DB01946
|
3-[1-(3-Aminopropyl)-1h-Indol-3-Yl]-4-(1 ...
|
Drugbank
DB02010
|
|
Drugbank
DB04522
|
|
|
|
Comment
|
AKT1 is localized in brain.
|
Formal Description Interaction-ID: 1943
|
|
Drugbank entries
|
Show/Hide entries for
AKT1
|
Drugbank
DB00171
|
|
Drugbank
DB01169
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB07584
|
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)phe ...
|
Drugbank
DB07585
|
5-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-4 ...
|
Drugbank
DB00171
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
|
|
Comment
|
One possibility for the down-regulation of Akt activation in AD brain is direct inhibition mediated by an increase in cellular beta-amyloid.
|
Formal Description Interaction-ID: 1954
|
|
Drugbank entries
|
Show/Hide entries for
AKT1
|
Drugbank
DB00171
|
|
Drugbank
DB01169
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB07584
|
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)phe ...
|
Drugbank
DB07585
|
5-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-4 ...
|
Drugbank
DB00171
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
|
|
Comment
|
The association of beta-amyloid with each of Akt1 and PDK was increased in AD brain. Beta-amyloid has specific affinity for PDK/Akt.
|
Formal Description Interaction-ID: 1955
|
interacts (colocalizes) with
|
Drugbank entries
|
Show/Hide entries for
AKT1
|
Drugbank
DB00171
|
|
Drugbank
DB01169
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB07584
|
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)phe ...
|
Drugbank
DB07585
|
5-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-4 ...
|
Drugbank
DB00171
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
|
|
Comment
|
Ser473 phosphorylation is required for full Akt activity and precedes the phosphorylation of Thr308 by PDK-1.
|
Formal Description Interaction-ID: 1976
|
increases_phosphorylation of
at Thr308; phosphorylation at Ser473 is required for full Akt activity;
|
Drugbank entries
|
Show/Hide entries for
PDPK1
or
AKT1
|
Drugbank
DB00482
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB01933
|
|
Drugbank
DB01946
|
3-[1-(3-Aminopropyl)-1h-Indol-3-Yl]-4-(1 ...
|
Drugbank
DB02010
|
|
Drugbank
DB03777
|
|
Drugbank
DB04522
|
|
Drugbank
DB06932
|
10,11-dimethoxy-4-methyldibenzo[c,f]-2,7 ...
|
Drugbank
DB07033
|
5-HYDROXY-3-[(1R)-1-(1H-PYRROL-2-YL)ETHY ...
|
Drugbank
DB07132
|
1-{2-OXO-3-[(1R)-1-(1H-PYRROL-2-YL)ETHYL ...
|
Drugbank
DB07300
|
2-(1H-imidazol-1-yl)-9-methoxy-8-(2-meth ...
|
Drugbank
DB07456
|
3-(1H-INDOL-3-YL)-4-(1-{2-[(2S)-1-METHYL ...
|
Drugbank
DB07457
|
3-[1-(3-AMINOPROPYL)-1H-INDOL-3-YL]-4-(1 ...
|
Drugbank
DB00482
|
|
Drugbank
DB01933
|
|
Drugbank
DB01946
|
3-[1-(3-Aminopropyl)-1h-Indol-3-Yl]-4-(1 ...
|
Drugbank
DB02010
|
|
Drugbank
DB04522
|
|
Drugbank
DB00171
|
|
Drugbank
DB01169
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
Drugbank
DB07584
|
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)phe ...
|
Drugbank
DB07585
|
5-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-4 ...
|
Drugbank
DB00171
|
|
Drugbank
DB01863
|
Inositol 1,3,4,5-Tetrakisphosphate
|
|
|